Protein Details: Transient receptor potential cation channel subfamily M member 4

Protein ID

ICDB_Pro_1315

Protein Name

Transient receptor potential cation channel subfamily M member 4

Gene Name

TRPM4; LTRPC4

Organism

Homo sapiens (Human)

Length

1214 amino acids

AlphaFoldDB

AF-Q8TD43-F1-model_v4.pdb

Function

Sequence

MVVPEKEQSWIPKIFKKKTCTTFIVDSTDPGGTLCQCGRPRTAHPAVAMEDAFGAAVVTVWDSDAHTTEKPTDAYGELDFTGAGRKHSNFLRLSDRTDPAAVYSLVTRTWGFRAPNLVVSVLGGSGGPVLQTWLQDLLRRGLVRAAQSTGAWIVTGGLHTGIGRHVGVAVRDHQMASTGGTKVVAMGVAPWGVVRNRDTLINPKGSFPARYRWRGDPEDGVQFPLDYNYSAFFLVDDGTHGCLGGENRFRLRLESYISQQKTGVGGTGIDIPVLLLLIDGDEKMLTRIENATQAQLPCLLVAGSGGAADCLAETLEDTLAPGSGGARQGEARDRIRRFFPKGDLEVLQAQVERIMTRKELLTVYSSEDGSEEFETIVLKALVKACGSSEASAYLDELRLAVAWNRVDIAQSELFRGDIQWRSFHLEASLMDALLNDRPEFVRLLISHGLSLGHFLTPMRLAQLYSAAPSNSLIRNLLDQASHSAGTKAPALKGGAAELRPPDVGHVLRMLLGKMCAPRYPSGGAWDPHPGQGFGESMYLLSDKATSPLSLDAGLGQAPWSDLLLWALLLNRAQMAMYFWEMGSNAVSSALGACLLLRVMARLEPDAEEAARRKDLAFKFEGMGVDLFGECYRSSEVRAARLLLRRCPLWGDATCLQLAMQADARAFFAQDGVQSLLTQKWWGDMASTTPIWALVLAFFCPPLIYTRLITFRKSEEEPTREELEFDMDSVINGEGPVGTADPAEKTPLGVPRQSGRPGCCGGRCGGRRCLRRWFHFWGAPVTIFMGNVVSYLLFLLLFSRVLLVDFQPAPPGSLELLLYFWAFTLLCEELRQGLSGGGGSLASGGPGPGHASLSQRLRLYLADSWNQCDLVALTCFLLGVGCRLTPGLYHLGRTVLCIDFMVFTVRLLHIFTVNKQLGPKIVIVSKMMKDVFFFLFFLGVWLVAYGVATEGLLRPRDSDFPSILRRVFYRPYLQIFGQIPQEDMDVALMEHSNCSSEPGFWAHPPGAQAGTCVSQYANWLVVLLLVIFLLVANILLVNLLIAMFSYTFGKVQGNSDLYWKAQRYRLIREFHSRPALAPPFIVISHLRLLLRQLCRRPRSPQPSSPALEHFRVYLSKEAERKLLTWESVHKENFLLARARDKRESDSERLKRTSQKVDLALKQLGHIREYEQRLKVLEREVQQCSRVLGWVAEALSRSALLPPGGPPPPDLPGSKD

PDB Structures

Ligand Binding

1. DICL_CP

2. DICL_Pep

Binding Site

171;421;448;828;831;865;868

Disease

Progressive Familial Heart Block;Type Ib and Erythrokeratodermia Variabilis Et Progressiva

Location

Widely expressed with a high expression in intestine and prostate. In brain; it is both expressed in whole cerebral arteries and isolated vascular smooth muscle cells. Prominently expressed in Purkinje fibers. Prominently expressed in Purkinje fibers. Prominently expressed in Purkinje fibers. Expressed at higher levels in T-helper 2 (Th2) cells as compared to T-helper 1 (Th1) cells. Expressed in keratocytes. .

DOI ID

10.1073/pnas.191360198; 10.1016/s0092-8674(02)00719-5; 10.1016/s0960-9822(03)00431-7; 10.1074/jbc.m305127200; 10.1038/ng1285; 10.1101/gr.2596504; 10.1161/01.res.0000147311.54833.03; 10.1113/jphysiol.2004.063974; 10.1113/jphysiol.2004.070839; 10.1007/s00424-003-1221-x; 10.1126/science.1098845; 10.1074/jbc.m411089200; 10.1074/jbc.m501686200; 10.1074/jbc.m506965200; 10.1016/j.ceca.2006.04.032; 10.1038/sj.emboj.7600963; 10.1080/10799890600637506; 10.1124/mol.105.021154; 10.1016/j.bbrc.2009.11.142; 10.1002/jcp.22310; 10.4049/jimmunol.1000880; 10.1038/nature24674; 10.1126/science.aar4510; 10.1172/jci38292; 10.1161/circgenetics.109.930867; 10.1002/humu.21599; 10.1016/j.jid.2018.10.044

RefSeq

NP_001182156.1 [Q8TD43-3]; NP_001308212.1 [Q8TD43-2]; NP_060106.2 [Q8TD43-1]

Feature